The reduced folate/methotrexate carrier and a membrane-associated folate binding protein as transport routes for novel antifolates: structure-activity relationships

G Jansen, G R Westerhof, J H Schornagel, A L Jackman, F T Boyle

Research output: Contribution to journalArticleAcademic

5 Citations (Scopus)
Original languageEnglish
Pages (from-to)767-70
Number of pages4
JournalAdvances in experimental medicine and biology
Volume338
Publication statusPublished - 1993

Keywords

  • Animals
  • Biological Transport
  • Carrier Proteins/metabolism
  • Folate Receptors, GPI-Anchored
  • Folic Acid Antagonists/metabolism
  • Kinetics
  • Leukemia L1210/metabolism
  • Mice
  • Quinazolines/chemistry
  • Receptors, Cell Surface/metabolism
  • Structure-Activity Relationship
  • Thymidylate Synthase/antagonists & inhibitors
  • Tumor Cells, Cultured

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